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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T14494 | Balovaptan | RG7314 | Vasopressin Receptor |
Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism. | |||
T4355 | Fuscoside | OPC 21268 | Vasopressin Receptor |
Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist. | |||
T6288 | Mozavaptan | OPC31260l,OPC-31260 | Vasopressin Receptor |
Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively. | |||
T64174 | Vasopressin V2 receptor antagonist 1 | ||
Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD). | |||
T11857 | LIT-001 | Oxytocin Receptor | |
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin receptor agonist with EC50 of 55 nM and Ki of 226 nM. | |||
T13920L | Terlipressin Acetate | Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous | Vasopressin Receptor |
Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelial cells (IEC-6).Terlipressin acetate exerts anti-in... | |||
T4141 | RG7713 | RO 5028442 | Vasopressin Receptor |
RG7713 (RO 5028442) has been used in trials studying Autistic Disorder. | |||
T5148 | Atosiban acetate | RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164 | Oxytocin Receptor , Vasopressin Receptor |
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban acetate (RW22164) inhibits... | |||
T7303 | LIXIVAPTAN | VPA-985,WAY-VPA 985 | Vasopressin Receptor |
Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM) | |||
T6453 | Conivaptan hydrochloride | Vaprisol,Conivaptan HCl,YM 087 | Vasopressin Receptor |
Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic. | |||
T2326 | Tolvaptan | OPC-41061 | Vasopressin Receptor , Autophagy |
Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia. | |||
T7434 | Argipressin | Arg8-vasopressin,Vasopressin,AVP | Vasopressin Receptor |
Argipressin (Vasopressin) is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth ... | |||
T2568 | Felypressin | Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2 | Vasopressin Receptor |
Felypressin (Octapressin) is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activity. | |||
T2568L | Felypressin acetate | 2-(L-Phenylalanine)-8-L-lysinevasopressin,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2 | Vasopressin Receptor |
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures. | |||
T4996 | Atosiban | RWJ22164,RW22164 | Oxytocin Receptor , Vasopressin Receptor |
Atosiban (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban inhibits the oxytocin-mediated rel... | |||
T21308 | Histrelin | Supprelin LA,Histrelin Acetate | Others |
Histrelin (Supprelin LA) acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It is considered a GnRH agonist. Histrelin is used in the treatment of hormone-sensitive cancers of th... | |||
T28153 | Nelivaptan | SSR149415,SR 149415,SR-149415 | Vasopressin Receptor |
Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist. | |||
T7284 | Argipressin acetate (113-79-1(free base)) | Others | |
Vasopressin acetate is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle... | |||
T15682 | L-371,257 | Oxytocin Receptor , Vasopressin Receptor | |
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a. | |||
T15273 | Fedovapagon | VA483,A106483 | Vasopressin Receptor |
Fedovapagon (VA106483) is a selective and potent agonist of the vasopressin V2 receptor (V2R) that inhibits the growth of intersegmental vessels in zebrafish. Fedovapagon can be used to study overactive bladder, nocturia... |